203888. lajstromszámú szabadalom • Eljárás pirazolo-piridin-gyűrűt tartalmazó mevalonsavszármazékok és ezeket hatóanyagként tartalmazó gyógyászati készítmények előállítására
1 HU 203 888 B 2 I. táblázat OH ( I - 2 ) R1 R2 R3 RJ H 2-Ph 4-F i-Pr H 1-Me 4-F i-Pr H 2-Me 4-F i-Pr H 1-i-Pr 4-F i-Pr H 1-t-Bu 4-F i-Pr H l-(4-MeO-Ph) 4-F i-Pr H 1-CHjPh 4-F i-Pr Me 2-Me 4-F i-Pr Me 1-Et 4-F i-Pr Me 1-i-Pr 4-F i-Pr Me l-(2’-piridil) 4-F i-Pr Et 1-Me 4-F i-Pr Et 1-Et 4-F i-Pr Et 1-i-Pr 4-F i-Pr Et 1-Ph 4-F i-Pr ciklo-Pr 1-Et 4-F i-Pr ciklo-Pr 1-i-Pr 4-F i-Pr ciklo-Pr 1-t-Bu 4-F i-Pr i-Pr 1-Me 4-F i-Pr i-Pr 2-Me 4-F i-Pr i-Pr 1-Et 4-F i-Pr i-Pr 1-i-Pr 4-F i-Pr i-Pr 1-t-Bu 4-F i-Pr i-Pr 2-Ph 4-F i-Pr i-Pr 1-Ph 4-F i-Pr t-Bu 1-Me 4-F i-Pr t-Bu 2-Me 4-F i-Pr t-Bu 1-Et 4-F i-Pr t-Bu 1-i-Pr 4-F i-Pr t-Bu 1-t-Bu 4-F i-Pr t-Bu 1-Ph 4-F i-Pr Ph 1-Et 4-F i-Pr Ph 1-i-Pr 4-F i-Pr Ph 1-t-Bu 4-F i-Pr Ph 1-Ph 4-F i-Pr 4-Cl-Ph 1-Et 4-F i-Pr 4-Cl-Ph 1-Ph 4-F i-Pr H 1-Ph 4-C1 i-Pr H 1-Me 4-C1 i-Pr H 1-Et 4-C1 i-Pr H 1-i-Pr 4-C1 i-Pr H 1-t-Bu 4-C1 i-Pr H 1-Ph 4-C1 i-Pr H l-(4-MeO-Ph) 4-C1 i-Pr H l-CH2Ph 4-C1 i-Pr R1 R2 R3 R3 Me 1-Me 4-C1 i-Pr Me 1-Et 4-C1 i-Pr Me 1-i-Pr 4-C1 i-Pr Me l-(4-MeO-Ph) 4-C1 i-Pr Me 1-t-Bu 4-C1 i-Pr Me 1-Ph 4-C1 i-Pr Me l-CHjPh 4-C1 i-Pr Me l-(2’-piridil) 4-C1 i-Pr Et 1-Me 4-C1 i-Pr Et 1-Et 4-C1 i-Pr Et 1-i-Pr 4-C1 i-Pr Et 1-Ph 4-C1 i-Pr ciklo-Pr 1-Me 4-C1 i-Pr ciklo-Pr 1-Et 4-C1 i-Pr ciklo-Pr 1-i-Pr 4-C1 i-Pr ciklo-Pr 1-t-Bu 4-C1 i-Pr i-Pr 1-Me 4-C1 i-Pr i-Pr 1-Et 4-C1 i-Pr i-Pr 1-i-Pr 4-C1 i-Pr i-Pr 1-t-Bu 4-C1 i-Pr i-Pr 1-Ph 4-C1 i-Pr t-Bu 1-Me 4-C1 i-Pr t-Bu 1-Et 4-C1 i-Pr t-Bu 1-i-Pr 4-C1 i-Pr t-Bu 1-t-Bu 4-C1 i-Pr t-Bu 1-Ph 4-C1 i-Pr Ph 1-Et 4-C1 i-Pr Ph 1-i-Pr 4-C1 i-Pr Ph 1-t-Bu 4-C1 i-Pr Ph 1-Ph 4-C1 i-Pr 4-Cl-Ph 1-Me 4-C1 i-Pr 4-Cl-Ph 1-Et 4-C1 i-Pr 4-Cl-Ph 1-Ph 4-C1 i-Pr H 1-Ph 4-F c-Pr H 2-Ph 4-F c-Pr H 1-Me 4-F c-Pr H 2-Me 4-F c-Pr H 1-Et 4-F c-Pr H 1-i-Pr 4-F c-Pr H 1-t-Bu 4-F c-Pr H l-(4-MeO-Ph) 4-F c-Pr H 1-CHiPh 4-F c-Pr Me 2-Me 4-F c-Pr Me 1-Et 4-F c-Pr Me 1-i-Pr 4-F c-Pr Me l-(4-MeO-Ph) 4-F c-Pr Me 1-Ph 4-F c-Pr Me 2-Ph 4-F c-Pr Me 1-CHjPh 4-F c-Pr Me l-(2’-piridil) 4-F c-Pr Et 1-Me 4-F c-Pr Et 1-Et 4-F c-Pr Et 1-i-Pr 4-F c-Pr Et 1-Ph 4-F c-Pr ciklo-Pr 1-Me 4-F c-Pr ciklo-Pr 1-Et 4-F c-Pr ciklo-Pr 1-i-Pr 4-F c-Pr 5 10 15 20 25 30 35 40 45 50 55 60 5
