193799. lajstromszámú szabadalom • Eljárás 3-acil-amino-metil-imidazo/1,2-a/piridin származékok és az ezeket a vegyületeket tartalmazó gyógyszerkészítmények előállítására
19379') 5 6 Táblázat (folytatás) Vegyület Y X Rí r2 Olvadáspont / 17.-ch 3 Cl 11-C4H9 ch3 182-183 18.-ch 3 Cl ch2c6h5 ch3 149-150 19.-ch 3 Cl-ch3 C2Hs 210-212 20.-ch 3 Cl-ch3 n-C3H7 193-195 21.-ch 3 Cl-ch3 i-C3H7 152-154 22. /2 .pd./-ch3 Cl-ch3 n-Ci+Hg 158-160 23.-ch 3 Cl-ch3 t—Ci*H 9 160-162 24.-ch 3 Cl-CH'3 c6h5 198-199 25. /5.pd. !-ch3 Cl-/CH 2 / 3 -186-187,5 26.-ch 3 Cl -/CH2 / j*-145-146 27.-ch 3 Cl-/CH 2/5-150-151 28.-ch 3 Cl-ch3 185-186 29.-ch 3 Cl-ch3 11-C5H11 127-129 30.-ch 3 Cl-ch3 a képlet 178-180 31 .-ch 3 Cl-ch3 n-CeHi3 104-105 32.-ch 3 Cl-ch3-CH2C6H5 126-127 33.-ch 3 Cl-ch3-CH-CHCH3 225-227 34.-ch 3-OCR 3-ch3 Tt-C3H7 135-136 35.-ch 3-och3-CII3 l—Ci+Hg 93-95 36.-ch 3-NO 2-ch3 n—C 3II7 154-156 37.-ch 3-no2-ch3 Í-C4H9 157-159 38.-ch 3-so2ck3-ch3 n-C3H7 182-183 39.-ch 3-so2ch3-ch3 Í-C9H9 120-122 40.-ch 3 11-ch3 n—C3II7 125-126,5 41 .-ch 3 H-ch3 i—Ci+Hg 154-156 42.-ch 3-nhcoch3-ch3 n-C3H7 110-111 43.-ch 3-nhcoch3-ch3 í —Ci*Hg 183-185 44.-ch 3-N/COCH3/2-ch3 n-C3H7 117-118 45.-ch 3-nh2-ch3 i—CgHg 177,5-178,5 46.-ch 3-nhch3-ch3 í—Ci*Hg 176-177 47.-ch 3-n/ch3/2-CHs i-C^Hg 117-118 48.-ch 3 Cl-ch3 4-Cl-CeHg 175-177 49.-ch 3 n-C 1*119-ch3 l‘”Cí+Hg 72,5-73 50.-ch 3-c2h5-ch3 Í—Ci+Hg 99-101 51 .-ch 3-c2h5-ch3 n-C3H7 108-110 52.-ch 3 F-CHs i“C i+H 9 184-185 53.-ch 3 F-ch3 n-C3H7 157-158 54.-ch 3-sch3-ch3 i—C9H9 102-104 55.-ch 3-SCH 3-ch3 n-C3H7 128-129 56.-ch 3-CH 3-ch3 Í-Cí+Hg 129-131 57.-ch 3-CH 3-ch3 n—C3H7 145-147 58. R Cl-ch3 i“CgH 9 90-91 59. H Cl-ch3 n-C3H7 171-173 60. Cl Cl-ch3 3_—Cl*H g 176-177 61 . Cl Cl-CHs n-C3H7 188-189 62. Cl F-ch3 n-C3H 7 154-155 63. Cl F-ch3 í-CifHg 173-174 64. Cl-C2H5-ch3 n—C 3H7 134-136 65. Cl-C2Hs-ch3 i-Ci+H 9 111-112 66. Cl-ch3-ch3 n-C3H7 164-165 67. Cl-ch3-CIÎ3 i—Ci*Hg 154-155 68. Cl-och3-ch3 n-C3H7 152-153 69. Cl-OCR 3-ch3 i—Ci*Hg 131-132 70. Cl-sella-ch3 TI-C3H7 139-141 71. Cl-sch3-CHs Í-C4H9 135-136 4
