199159. lajstromszámú szabadalom • Eljárás véralvadásgátló peptidek és ezeket hatóanyagként tartalmazó gyógyszerkészítmények előállítására

199159

12

21. példa

H-Gly-Asp-Phe-Glu-Glu-Ile-NMePgl-Glu--Glu-íyr-Leu-Gln-OH

22. példa

H-Gly-Asp-Phe-Glu-Pro-Ile-Pro-Glu-Asp-Ala-Tyr-Asp-Glu-OH

23. példa

H-Ser-His-Asn-Asp-Gly-Asp-Phe-Glu-Glu-Ile-Pro-Glu-Glu-Tyr-Leu-Gtn-OH

24. példa

H-Gly-Asp-Phe-Glu-Pro-Ile-Pro-Glu-Asp-Ala-Tyr-Pco-NH2

25. példa

Suc-Phe-Glu-Pro-Ile-Pro-Glu-Asp-Ala-Tyr-Pro-NH2

26. példa

H-Asp-Phe-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Tyr-Gln-OH

27. példa

H-Asp-Phe-Glu-Glu-lle-Pro-Glu-Glu-Ala-Tyr-Gln-OH

28. példa

H-Asp-Phe-Glu-Glu-Ile-Pro-Glu-Asp-Ala-Tyr-Gln-OH

2d példsi

Suc-Phe-Glu-Pro-Ile-Pro-Glu-Glu-Tyr-Leu-Pro-NH2

30. példa

H-Gly-Asp-béta-(2-tienil)-alanil-Glu-Glu-Ile-Pro-Glu-Glu-Tyr-Leu-Gln-OH

31. példa

H-Gly-Ala-O-metil-tirozil-Glu-Glu-Ile-Pro-Glu-Glu-Tyr-Leu-GIn-OH

32. példa

Suc-Phe-Glu-Pro-lle-Pro-Glu-Glu-Pro-OH

33. példa

H-Asp-Phe-Glu-Glu-lle-Pro-Glu-Ala-Tyr--Leu-Gln-OH

34. példa

H-Asp-Phe-Glu-Glu-Ile-Pro-Glu-Glu-Ala-Leu.-Gln-OH

35. példa

H-Gly-Asp-Phe-Glu-Glu-Leu-Pro-Glu-Glu-Tyr-Leu-Gln-OH

36. példa

H-Gly-Asp-Phe-Glu-Glu-Val-Pro-Glu-Glu-Tyr-Leu-Gln-OH ’

37. példa

H-Gly-Asp-Phe-Glu-Glu-Phe-Pro-Glu-Glu - -Tyr-Leu-uln-OH

38. példa

H-Asp-Phe-Glu-Pro-Ile-Pro-Glu-Glu-Tyr-Leu-Gln-OH

39. példa

Suc-Phe-Glu-Pro-Ile-Pro-Glu-Glu-Tyr-Leu-Gln-OH

11

40. példa

H-Gly-Asp-Phe-Glu-Pro-IIe-Pro-GIu-Asp-Ala-Tyr-Glu-OH

41. példa

H-Gly-Asp-Phe-Glu-Glu-Ile-Pro-Glu-Asp-Ala-Phe-Asp-Glu-OH

42. példa

Ac-Phe-Glu-Glu-Ile-Pro-Glu-Glu-Tyr-Leu - -Orn-NH2

43. példa

H-Gly-Asp-Phe-Glu-Pro-Ile-Pro-Glu-Glu-Tyr-Tyr-Glu-OH

44. példa

H-Asp-Phe-Glu-Pro-Ile-Pro-Glu-Glu-Tyr-Tyr-Gln-OH

45. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Phe-Lys-NH2

46. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Phe-D-Lys-NH2

47. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Phe-Orn-NHj

48. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Ala-Tyr-Lys-NH2

49. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Phe-Lys-ÖH

50. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-His'-Lys-OH

51. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Cha-Lys-NH2

52. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Leu-Phe-Lys-NH2

53. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Gln-Glu-Ala-Phe-Lys-NH2

54. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Phe-Glu-OH

55. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Phe-Gln-OH

56. példa

Suc-Tyr-Glu-Pro-Ile-Pro-Glu-Glu-Ala-Cha-Asp-OH

57. példa

H-Gly-Asp-Phe-Glu-Pro-Ile-Pro-Glu-Asp-Ala-Tvr-D-Asn-OH

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