195476. lajstromszámú szabadalom • Eljárás alfa-amino-alkil-alfa-alkil-fenil-acetonitril származékok és az ilyen hatóanyagot tartalmazó gyógyászati készítmények előállítására
195 476 V. táblázat folytatása példa száma R1 R2 R3 111 n R4 R5 R6 R7 69. 3 -Omc 4-OMe H 3 2 iPr Me 3-Me 4-C! 70. 3-OMe 4-OMe H 3 2 iPr H 3-OMe 4-OMe 71. 3-OMc 4-OMc H 3 3 iPr H 4-F H 72. 3-OMe 4-OMe H 3 3 iPr Me 4-F H 73. 3-OMc 4-OMe H 3 3 iPr H 2-OMe H 74. 3-OMe 4-OMe H 3 3 iPr Me 2-OMe H 75. 3-OMe 4-OMe H 3 3 Me H 4-F H 76. 3-OMe 4-OMe H 3 3 Me Me 4-F H 77. 3-OMe 4-OMe 5-OMe 2 2 iPr Me H H 78. 3-OMe 4-OMe 5-OMe 2 2 iPr H 2-OMe H 79. 3-OMe 4-OMe 5-OMe 2 2 iPr Me 2-OMe H 80. 3-OMe 4-OMe 5 -OMe 2 3 Me H 2-OMe H 81. 3-OMe 4-OMe 5-OMe 2 3 Me Me 2-OMe H 82. 3-OMe 4-OMe 5-OMe 2 3 Et H 2-OMe H 83. 3-OMe 4-OMe 5-OMe 2 3 Et Me 2-OMe H 84. 3-OMe 4-OMe 5-OMe 2 3 nPr H 2-OMe H 85. 3-OMe 4-OMe 5-OMe 2 3 nPr Me 2-OMe H 86. 3-OMe 4-OMe 5-OMe 2 3 nBu H 2-OMe H 87. 3-OMe 4-OMe 5-OMe 2 3 nBu Me 2-OMe H 88. 3-OMe 4-OMe 5-OMe 2 3 iBu H 2-OMe H 89. 3-OMe 4-OMe 5-OMe 2 3 iBu Me 2-OMe H 90. 3-OMe 4-OMe 5-OMe 3 2 iPr Me H H 91. 3-OMe 4-OMe 5-OMe 3 2 iPr H 4-F H 92. 3-OMe 4-OMe 5-OMe 3 2 iPr Me 4-F H 93. 3-OMe 4-OMe 5-OMe 3 2 iPr H H-Cl H 94. 3-OMe 4-OMe 5-OMe 3 2 iPr Me 4-C1 H 95. 3-OMe 4-OMe 5-OMe 3 2 iPr H 3-Me H 96. 3-OMe 4-OMe 5-OMe 3 2 iPr Me 3-Me H 97. 3-OMe 4-OMe 5-OMe 3 2 iPr H 2-Me H 98. 3-OMe 4-OMe 5-OMe 3 2 iPr Me 2-Me H 99. 3-OMe 4-OMe 5-OMe 3 2 iPr H 3-OMc H 100. 3-OMe 4-OMe 5-OMe 3 2 iPr H 2-OMe H 101. 3-OMe 4-OMe 5-OMe 3 2 iPr Me 2-OMe H 102. 3-OMe 4-OMe 5-OMe 3 2 iPr H 2-OMe 6-OMe 103. 3-OMe 4-OMc 5-OMe 3 2 iPr H 2-OEt H 104. 3-OMc 4-OMe 5-OMe 3 2 Me H 2-OMe H 105. 3-OMe 4-OMe 5-OMe 3 2 Me Me 2-OMe H 106. 3-OMc 4-OMe 5-OMe 3 2 Et H 2-OMe H 107. 3-OMe 4-OMe 5-OMe 3 2 nPr H 2-OMe H 108. 3-OMe 4-OMe 5-OMe 3 2 nBu H 2-OMe H 109. 3-OMe 4-OMe 5-OMe 3 2 iBu H 2-OMe H 110. 3-OMe 4-OMe 5-OMe 3 3 iPr H H H 111. 3-OMc 4-OMe 5-OMe 3 3 iPr Me H H 112. 3-OMe 4-OMe 5-OMe 3 3 iPr H 4-F H 113. 3-OMe 4-OMe 5-OMe 3 3 iPr Me 4-F H 114. 3-OMc 4-OMe 5-OMe 3 3 iPr H 3-F H 115. 3-OMe 4-OMe 5-OMe 3 3 iPr Me 3-F H 116. 3-OMe 4-OMe 5-OMe 3 3 iPr H 2-F H 117. 3-OMe 4-OMe 5-OMe 3 3 iPr Me 2-F H 118. 3-OMe 4-OMe 5-OMe 3 3 iPr H 4-C1 H 119. 3-OMe 4-OMe 5-OMe 3 3 iPr Me 4-C1 H 120. 3-OMe 4-OMe 5-OMe 3 3 iPr H 3-C1 H 121. 3-OMe 4-OMc 5-OMe 3 3 iPr Me 3-C1 H 122. 3-OMe 4-OMc 5-OMe 3 3 iPr H 2-C1 H 123. 3-OMe 4-OMe 5-OMe 3 3 IPr Me 2-C1 H 124. 3-OMe 4-OMe 5-OMe 3 3 iPr H 4-Me H 125. 3-OMe 4-OMe 5-OMe 3 3 iPr Me 4-Me H 126. 3-OMe 4-OMe 5-OMe 3 3 iPr H 3-Me H 127. 3-OMe 4-OMe 5-OMe 3 3 iPr Me 3-Me H 128. 3-OMe 4-OMe 5-OMe 3 3 iPr H 2-Me H 3
