179259. lajstromszámú szabadalom • N-szubsztituált Ó-aminosavak előállítására

179259 6 A találmány szerinti eljárással előállított hatóanyagok és olvadáspontjuk. 1. táblázat A vegyü­let R sorszáma R1 R2 R3 R4 X Y z Op. °r 1 CH3-CH3-CH(CH3)­H H H H Cl H H 122 2 CH3-C(CH3)2-H H H H Cl H H 166 3 CH3-CH2-CH(CH3)­H ch3 H H a H H 95 4 c6h,,­H ch3 6—CH3 H Cl H H 103 5 ch3-ch2-H ch3 6—CH3 H Cl H H 101 6 ch3-H ch3 6-C2Hs H ci H H 123 7 ch3-ch2~ch2-H ch3 6—CH3 H Cl H H 125 8 CH3-C(CH3)2-H ch3 6-CH3 H a H H 162 9 ch2=ch-ch2-H ch3 6-CH3 H Cl H H 131 10 c2h5— H ch3 6—C2Hs H Cl H H 78 11 ch3-ch2-ch2-H ch3 6—C2Hs H a H H 129 12 CH3-CH-(CH3)­H ch3 6-C2Hs H Cl II H 135 13 ch3-ch2-ch2-ch2-H ch3 6—C2Hs H a H H 112 14 CH3-CH2-CH(CH3)­H ch3 6-C2Hs H Cl H H 98 15 CH3-C(CH3)2-H ch3 6-C2Hs H a H H 75 16 CH3-CH(CH3)-CH2-H ch3 6—C2H5 H a H H 153 17 CH3-(CH2)3-CH2-H ch3 6—C2Hs H Cl H H 55 18 CH3-(CH2)4-CH2-H ch3 6—C2H5 H Cl H H 60 19 CH3OCH2-CH2-CH3-H ch3 6—C2Hs H Cl H H 80 20 ch2=ch-ch2-H ch3 6—C2Hs H Cl H H 123 21 c6h,,­H ch3 6-C2Hs H a H H 145 22 ch3-H c2h5 6—C2H5 H Cl H H 134 23 ch3-ch2-H c2h5 6—C2H5 H Cl H H 128 24 ch3-ch2-ch2-H c2h5 6—C2Hs H ci H H 123 25 CH3-CH2-CH2-ch3 C2Hs 6—C2Hs H Cl H H 120 26 CH3-CH(CH3)­H C2Hs 6—C2Hs H a H H 126 27 CH3-CH2-CH(CH3)­H C2Hs 6—C2H5 H Cl H H 72 28 CH3-CH(CH3)-CH2-H c2h5 6—C2 Hs H a H H 85 29 CH3-CH(CH3)-CH2-ch3 c2h5 6-C2Hs H a H H 113 30 ch2=ch-ch2-H c2h5 6—C2 Hs H a H H 110 31 ch2=ch-ch2-ch3 C2Hs 6—C2 Hs H a H H 128 32 CH3OCH2-CH2-CH2-H c2h5 6—C2Hs H ci H H 97 33 oh-ch2-ch2-H c2h5 6—C2Hs H Cl H H 44-45 34 oh-ch2-ch2-H c2h5 6—C2H5 H a Cl H 50-55 35 oh-ch2-ch2-H ch3 6—CH3 H a Cl a 105-110 36 ch3-H ci H H a H H 111 37 ch3-ch2-H Cl H H a H H 70 38 CH3-CH2-CH(CH3)­H a H H a H H 55 39 ch3och2-CH2-CH2-H a H H a H H 29 40 CH2=CH-CH2-H Cl H H ci H H 44 41 CH3-CH(CH3)­H H H 4—Cl Cl H H 160 42 c6h,,­H H H 4—Cl Cl H H 175 43 ch3-ch2-H H 3—Cl 4—Cl a H H 137 44 CH3-CH2-CH2-H H 3—Cl 4—Cl a H H 152 45 c6h, H no2 H H a H H 100 46 ch3-ch2-ch2-H H 3—N02 H a H H 52 47 c6h„­H H 3—N02 H a H H 92 48 CH3-CH2-CH(CH3)­H H H H a a H 125 49 CH3-CH2-CH(CH3)­H ch3 H H a Cl H 132 50 ch3-H ch3 6—CH3 H Cl a H 157 51 ch3-ch2-H ch3 6-CH3 H a a H 159 52 ch3-ch2-ch2-H ch3 6-CH3 H a Cl H 140 53 ch3-C(ch3)2-H ch3 6-CH3 H a a H 143 54 ch2=ch-ch2-H ch3 6-CH3 H ci Cl H 1 ly 55 ch3-ch2-H ch3 6-C2 Hs H ci a H 138 3

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