167158. lajstromszámú szabadalom • Eljárás 6-[alfa-imidoilaminoalkanoilamino]-aracil- amino penám-3-karbonsavak előállítására

27 167158 28 Ar Rí R2 R5 Cfi

H 6"S C6

H

5 C6

H

5

QU,— C6

H

5

QHS

C6

H

5

C6

H

S

C6

H

5

C6

H

5

C6

H

S

C6

H

5

C6

H

5

QH5

C6

H

5

C6

H

5

-4-HOC6

H4-4-HOC6

H4-4-H0QH4-4-H0QH4-4-HOC6

H4-4-H0C6

H4-4-HOC6

H4-4-HOQH4-4-HOC6

H4-I CH3CHI CH3CH-CH2

-CH2

-CH2

-CH2

I CH3 CH2 CH— -CH2

I CH3CH-CH2

-CH2

I CH3CHI CH3CHI CH3 CH2 CH— -CH2

-CH2

-CH2

-CH2

I CH3 CH2 CH-CH2

I CH3CHI CH3CHI CH3 CH2 CH— -CH2

I CH3CHCH3

HHHC2

H

5

— HH-i-C3

H

7

HCH3

HCH3

CH3-CH3

CH3

n-C3

H

7

C2

H

S

HHCH3

HHHHCH3-CH, p-<CH3)2

NC

6

H4-HP-0C6

H4. CH3

m-0C6

H4-n-C3

H

7

m-NCC6

H4-H- m-NCC6

H4-H- o-HOC6

H4-CH3

p-HOC6

H4-H- p-HOC6

H

4

H- p-CH3

CONHC

6

H4-CH3

p-CH3

C0NHC

6

H4-H- p-C2

H

s

CONHC

6

H4 C2

H

5

— p—CH3 SCg H4

— C2

H

5

p—CH3

S0

2

C

6

H4

— H- m-H2

NS0

2

C

6

H4-CH3

p-CH3

NHS0

2

C

6

H4-H- m-(CH3

)

2

NS0

2

C

6

H4-H- p-CH3

COC

6

H4-H- m-CH3

COC

6

H4-H- m-CH3

C0C

6

H4-CH3

p-(CH3

)

2

NC

6

H4-HP-0QH4-n-C3

H

7

m-NCC6

H4-CH3 HC2

H

S

— p-HOC6

H4-p-CH3

C0NHC

6

H4-p—CH3

S0

2

Cg H4 -i4